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1º PARCIAL DE BIOFARMACIA Y FARMACOCINETICA GRUPOS C Y D
CURSO 2004-2005
Un fármaco se administra vía intravenosa, con una dosis de 400 mg y se observa una disminución de concentraciones plasmáticas desde 150 mg/l hasta 75 mg/l durante un tiempo de 2 horas. Calcule el tiempo necesario para una concentración terapéutica mayor o igual a 10 mg/l. Vd= 15l
Sabiendo las constantes cinéticas de un fármaco, calcule la semivida biologica. Datos: k12= 0.05h-1 , k21= 0.08h-1 , k13= 0.43h-1 , = 0.5h-1
Complete:
At= C+P+……
….=D/(C0/kel)
el=k13….."Cdt
C"=…./kel*Vd
Un fármaco, vía intravenosa se sabe que se ha administrado a una dosis de 200 mg y que su vd=20L y tiene un Cl=1L/h. El mismo fármaco se administra vía intravenosa a una dosis de 600 mg. Calcule la semivida biológica, C0 y AUC.
Para un fármaco se conoce un Clt=1L/min. Tras la administración de una dosis de 100 mg intravenosa. Se recoge en orina 25 mg de fármaco al pasar 9t1/2. A partir de esta información puede calcular Clh?
Tras una dosis de 200 mg intravenosa, tras 4 horas se recogen 15 mg de fármaco, ¿se puede calcular el aclaramiento renal?
¿Cuál es el aclaramiento hepático óptimo de un fármaco para un individuo sano?
Tras la administración intravenosa de una dosis de 200 mg se obtiene la siguiente curva: C0 30e-0.2t. Calcule C".La velocidad de perfusión es de 0.1 g/h. ¿Qué tiempo pasara hasta alcanzar el 95% del estado estacionario?
Tras la administración intravenosa, se recoge orina y se ve que apenas hay fármaco. ¿Es que no se ha filtrado a nivel glomerular?
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Enviado por: Sheila Idioma: castellanoPaís: España